Publications

132.  Safer, Greener, and more Facile Alternatives for Synthesis of Organic Azides. Sebeika, M.M.; Jones, G.B. Current Organic Synthesis. 2014. Epub, Ahead of Print.
131. Accelerated Labeling Methods and Syntheses of Radiotracers Utilizing Microfluidic Technology. Hargrove, K.; Jones, G.B. Current Radiopharmaceuticals. 2014. Epub, Ahead of Print.
130. Hypoxia-induced and A2A adenosine receptor-independent T-cell suppression is short lived and easily reversible. Ohta, A.; Madasu, M.; Subramanian, M.; Kini, R.; Jones, G.; Chouker, A.; Ohta, A.; Sitkovsky, M. International Immunology. 2014, 26, 83-91.
129. Design and evaluation of xanthine based adenosine receptor antagonists: Potential hypoxia targeted immunotherapies. Thomas, R.; Lee, J.; Chevalier, V.; Sadler, S.; Selesniemi, K.; Hatfield, S.; Sitkovsky, M.; Ondrechen, M. J.; Jones, G. B. Bioorganic & Medicinal Chemistry. 2013, 21, 7453-7464.
128. Fluoroalkynylations of Aryl Halides under Continuous-Flow Homogeneous Catalysts. Placzek, M.S.; Chmielecki, J.M.; Houghton, C.; Calder, A.; Wiles, C.; Jones, G.B. J. Flow Chem. 2013, 3(2), 46-50.
127. Extending the versatility of the Hemetsberger-Knittel indole synthesis through microwave and flow chemistry. Ranasinghe, N.; Jones, G. B., Bioorg. Med. Chem. Lett. 2013, 23(6), 1740-1742.
126. Microwave and continuous flow technologies in drug discovery. Sadler, S.; Moeller, A.R.; Jones, G.B. Expert Opinion in Drug Discovery2012, 7(12), 1107-1128.

125. The Forward Path for Biopharmaceuticals and Biosimilars: Emerging Options in the Selection of Host Cell Systems. Wager, K.; Jones, G.B. Current Biotechnology. 2012, 1(4), 297-317.

124.   Analytical tools for characterizing biopharmaceuticals and the implications for biosimilars.  Berkowitz, Steven A.; Engen, John R.; Mazzeo, Jeffrey R.; Jones, Graham B. Nature Reviews Drug Discovery, 2012, 11, 527-540.

123.   Synthesis and evaluation of potent and selective human V1a receptor antragonists as potential ligands for PET or SPECT imaging. Fabio, Karine; Guillon, Christophe; Lacey, Carl J.; Lu, Shi-fang; Heindel, Ned D.; Ferris, Craig F.; Placzek, Michael; Jones, Graham; Brownstein, Michael J.; Simon, Neal G. Bioorganic and Medicinal Chemistry, 2012, 20, 1337-1345.

122.     Microwave Accelerated Labeling Methods in the Synthesis of Radioligands for Positron Emission Tomography Imaging, Kallmerten, Amy; Alexander, Abigail; Wager, Krista; Jones, Graham, Current Radiopharmaceuticals, 2011, 4 (4), 343-354

121.     Internalization of C17α-alkynylestradiol-porphyrin conjugates into estrogen receptor positive MCF-7 breast cancer cells, Sadler, Sara; Persons, Kelly S.; Jones, Graham B.; Ray, Rahul, Bioorganic and Medicinal Chemistry Letters, 2011, 21(15), 4638-4641.

120.     Microwave accelerated three-component fluoroalkylations: expeditious routes to fluoropharmaceuticals and PET ligands, Placzek, Michael; LaBeaume, Paul; Harris, Luke; Ng, Patrick; Daniels, Mathew; Kallmerten, Amy; Jones, Graham B., Tetrahedron Letters, 2011, 52, 332.

119.     An efficient route to xanthine based A2A adenosine receptor antagonists and functional derivatives, LaBeaume, Paul; Dong, Ma; Sitkovsky, Michail; Jones, Elizabeth V.; Thomas, Rhiannon; Sadler, Sara; Kallmerten, Amy E.; Jones, Graham B. Organic and Biomolecular Chemistry, 2010, 8, 4155.

118.     Radio-Iodination Methods for the Production of SPECT Imaging Agents, Wager, K., Jones, G.B., Current Radiopharmaceuticals, 2010, 3 (1) 37.

117.     Microwave Accelerated Synthesis of PET Image Contrast Agents for AD Research, Kallmerten A.E., Jones, Graham B., Current Alzheimer Research, 2010, 7, 251.

116.     Microwave-accelerated fluorodenitrations and nitrodehalogenations: expeditious routes to labeled PET ligands and fluoropharmaceuticals, LaBeaume, P.,  Placzek, M., Daniels, M., Kendrick, I., Ng,  P., McNeel, M.,  Afroze, R.,  Alexander, A., Thomas, R., Kallmerten, A.E., Jones, G.B., Tetrahedron Letters, 2010 51(14), 1906-1909.

115.  Synthesis, functionalization and photo-Bergman chemistry of enediyne bioconjugates, LaBeaume, P., Wager, K.,  Falcone, D.,  Li, J.,  Torchilin, V.,  Castro, C.,  Holewa, C. Kallmerten, A.E., Jones, G.B. , Bioorganic and Medicinal Chemistry. 2009  17 (17), 6292.

114. Designed DNA Probes from the Neocarzinostatin Family: Impact of Glycosyl Linkage Stereochemistry on Bulge Base Binding, Ma, D. ; Lin, Y. ;  Xiao, Z. ;   Kappen, L. ;   Goldberg, I. H. ; Kallmerten, A. E. ; Jones, G. B.  Bioorganic and Medicinal Chemistry2009, 17(6), 2428.

113. An Efficient Route to Novel A2A Adenosine Receptor Antagonists, Analogues and Prodrugs, Ma, D, Sitkovsky, M., Kallmerten, A.E., Jones, G.B. Tetrahedron Letters, 2008, 49, 4633.

112. Designed Molecular Probes of DNA Bulges:  Jones GB; Lin Y; Ma D; Xiao Z; Hwang G; Kappen L; Goldberg I. H. Current topics in medicinal chemistry 2008,  8,  436.

111. Photoactivated Enediynes as Targeted Antitumoral Agents: Efficient Routes to Antibody and Gold Nanoparticle Conjugates, Danielle Falcone, Jane Li, Amit Kale and Graham B. Jones, Bioorganic and Medicinal Chemistry Letters. 2008, 18, 934.

110. DNA Interactive Enediyne Antitumor Agents and their Congeners, Graham B. Jones and Danielle Falcone ed. M. Lee, in Synthetic and Biophysical Studies of DNA Binding Compounds, Lee, M.; Strekowski, L. Eds. 2007, Transworld Research, pp.169-196. ISBN: 978-81-7895-290-1.

109. Chiral Auxiliaries derived from Biogenic Building Blocks bearing h6 Arene Cr(0) Complexes, Jane Li, Longfei Xie, Mustafa Guzel, Steven B. Heaton, Amy E. Kallmerten and Graham B. Jones, Journal of Organometallic Chemistry. 2007, 692, 5459.

108. Solution Structure of a Designed Spirocyclic Helical Ligand Binding at a Two-Base Bulge Site in DNA. Zhang, Na; Lin, Yiqing; Xiao, Ziwei; Jones, Graham B.; Goldberg, Irving H. Biochemistry. 200746,  4793.

107. Solution Structure of a Designed Spirocyclic Helical Ligand Binding at a Two-Base Bulge Site in DNA, Na Zhang, Yiqing Lin, Ziwei Xiao, Graham B. Jones, and Irving H. Goldberg, Biochemistry2007, 46, 561.

106. Molecular Probes of DNA Bulges:  Functional Assay and Spectroscopic Analysis, Graham B. Jones, Yiqing Lin, Ziwei Xiao, Lizzy Kappen, and Irving H. Goldberg, Bioorg Med Chem2007, 15, 784.

105. Spirocyclic Helical Compounds as Binding Agents for Bulged RNA, Including HIV-2 TAR, Ziwei Xiao, Na Zhang, Yiqing Lin, Graham B. Jones, and Irving H. Goldberg, Chem Commun.  2006, 4431.

104. Nuclear Estrogen Recepter Targeted Photodynamic Therapy:  Selective Uptake and Killing of MCF-7 Breast Cancer Cells by a C17α-Alkynylestradiol-Porphyrin Conjugate, Swamy, N. ;  Purohit, A. ; Fernandez-Gacio, A. ; Jones, G. B. ; and Ray, R. ;  Journal of Cellular Biochemistry.  2006, 99, 966.

103. Microwave Expedited Synthesis of 5-Aminocamptothecin Analogs:  Inhimbitors of Hypoxia Inducible Factor HIF-1α, Joelle Torregrossa, Glenn J. Bubley, and Graham B. Jones, Bioorganic & Medicinal Chemistry Letters.  2006, 16, 6082-6085.

102. An Image contrast agent selectively activated by prostate specific antigen (PSA), Graham B. Jones, Curtis F. Crasto, Jude E. Matthews, Longfei Xie, Miguel O. Mitchell, Ahmed El-Shafey, Anthony V. D’Amico, and Glenn J. Bubley  Bioorganic and Medicinal Chemistry 2006, 14, 418.

101. Functionalized heterobifunctional poly[ethylene glycol] templates for use in cellular trafficking and imaging studies, Dinesh Shenoy, Wei Fu, Curtis Crasto, Srinivas Sridhar, Mansoor Amiji, Jane Li, James Weinberg, Graham Jones, Int. Journal of Nanomedicine, 2006, 1, 51.

100. Synthesis and Protein Degradation Capacity of Photoactivated Enediynes Fouad, F. S.; Wright, J. M.; Plourde, G., II.; Purohit, A. D.; Wyatt, J. K.; El-Shafey, A.; Hynd, G.; Crasto, C. F.; Lin, Y.; Jones, G. B. J. Org. Chem. 2005; 70, 9789.

99. An Approach to Heterobifunctional Poly(ethyleneglycol) Bioconjugates, Jane Li, Curtis F. Crasto, James Weinberg, Mansoor Amiji, Dinesh Shenoy, Srinivas Sridhar, Glenn Bubley, and Graham B. Jones, Bioorg. Med. Chem. Lett. 2005, 15, 5558.

98. Convenient synthesis of NCS-Chromophore metabolite isosteres: Binding agents for bulged DNA microenvironments, Yiqing Lin, Graham Jones, Geum-Sook Hwang, Lizzy Kappen, Irving Goldberg, Org. Lett. 2005, 7, 71.

97. Exploiting p Shielding Interactions: A Highly Selective Chiral Auxiliary derived from a Biogenic Building Block, Longfei Xie and Graham B. Jones, Tetrahedron Lett.  2005, 46, 3579.

96. Photoactivated Enediynes: targeted chimeras which undergo photo-Bergman cyclization, Farid S. Fouad, Curtis F. Crasto, Yiqing Lin and Graham B. Jones, Tetrahedron Lett.  2004, 45, 7753.

95. A Prospective, Multicenter, Randomized Phase II Trial of the Herbal Supplement, PC-SPES, and Diethylstilbestrol in Patients with Androgen-Independent Prostate Cancer, William K. Oh, Philip W. Kantoff, Vivian Weinberg, Graham Jones, Brian I. Rini, Mika K. Derynck, Robert Bok, Matthew R. Smith, Glenn J. Bubley, Robert T. Rosen, Robert S. DiPaola, Eric J. Small, J. Clin. Oncol. 2004, 22, 3705.

94. Preparation of Alkylation Agents for Bulged DNA Microenvironments, Farid S. Fouad, Zhen Xie, Irving H. Goldberg, and Graham B. Jones, Bioorganic and Medicinal Chemistry Letters 2004, 14, 3337.

93. A Practical method for preparation of b-glycosides of N-Acetylglucosamine, Curtis F. Crasto and Graham B. Jones, Tetrahedron Lett. 2004, 45, 4891.

92. Image contrast agents activated by prostate specific antigen (PSA), Graham B. Jones, Longfei Xie, Ahmed El-Shafey, Curtis F. Crasto, Glenn J. Bubley and Anthony V. D’Amico, Bioorganic and Medicinal Chemistry Letters 2004, 14, 3081.

91. Stereochemical Control of Small Molecule Binding to Bulged DNA: Comparison of Structures of Spirocyclic Enantiomer-Bulged DNA Complexes Hwang, G.-S.; Jones, G. B.; Goldberg, I. H.; Biochemistry, 2004, 43, 641.

90. Designed Enediyne Antitumor Agents, Graham B. Jones and Farid S. Fouad, Frontiers in Medicinal Chemistry, 2004, 1, 189-214.

89. The Photo-Bergman Cycloaromatization of Enediynes, Graham B. Jones and Keith C. Russell, CRC Handbook of Photochemistry, 2004, 29-1.

88. History of Anticancer Drugs, Jones, G.B.; eLS, 2003. Published online.

87. Solution structure of a wedge-shaped synthetic molecule at a two-base bulge site in DNA, Geum-Sook Hwang, Graham B. Jones, Irving H. Goldberg, Biochemistry, 2003, 42, 8472.

86. CYP2D6 – catalyzes tamoxifen aromatic hydroxylation with an NIH-Shift, Yiding Hu, Shangara S. Dehal, George Hynd, Graham B. Jonesand David Kupfer, Xenobiotica, 2003, 33, 141.

85. Stimulation of DNA strand slippage synthesis by a bulge binding synthetic agent, Lizzy S. Kappen, Zhen Xi, Graham B. Jones, Irving H. Goldberg, Biochemistry, 2003, 42, 2166.

84. Halo-Enediynes: Probing the Electronic and Stereoelectronic Contributions to the Bergman Cycloaromatization, Gary W. Plourde II, Philip M. Warner, Dennis A. Parrish, Graham B. Jones, Journal of Organic Chemistry,  2002, 67, 5727.

83. Oxa-Enediynes: Probing the Electronic and Stereoelectronic Contributions to the Bergman Cycloaromatization, Graham B. Jones, Justin M. Wright, George Hynd, Justin K. Wyatt, Philip M. Warner, Robert S. Huber, Aiwen Li, Michael W. Kilgore, Robert P. Sticca, and Richard S. Pollenz, Journal of Organic Chemistry,  2002, 67, 5369.

82. Protein Degradation with Photoactivated Enediyne-Amino Acid Conjugates, Gary Plourde, Ahmed El-Shafey, Farid, S. Fouad, Ajay S. Purohit, Graham B. Jones, Bioorganic and Medicinal Chemistry Letters 2002, 12, 2985.

81. Targeting DNA Bulged Microenvironments with Synthetic Agents: Lessons from a Natural Product, Zhen Xi, Guem-Sook Hwang, Irving H. Goldberg, Jeffrey L. Harris, William T. Pennington, Farid S. Fouad, Ghassan Qabaja, Justin M. Wright, Graham B. Jones, Chemistry & Biology, 2002, 9, 925.

80. Designed Enediyne Antitumor Agents, Graham B. Jones and Farid S. Fouad Current Pharmaceutical Design, 2002, 8, 2415.

79. Application of Affinity Capillary Electrophoresis for the Determination of Binding and Thermodynamic Constants of Enediynes with Bovine Serum Albumin and Histone H1, El-Shafey, A. ;  Zhong, H. ;  Jones, G. B. ; Krull, I. Electrophoresis 2002, 23, 945.

78. DNA Cleavage by Aromatic Amines, Jiwei Qi, Bin Meng, Gang Li, Philip M. Warner and Graham B. Jones, Bioorganic and Medicinal Chemistry Letters 2002, 12, 1.

77. Photoactivated Enediyne-Estrogens as Photochemical Proteases, Graham B. Jones, Ajay Purohit,Justin Wyatt, Narashima Swamy,and Rahul Ray, Tetrahedron Letters, 2001, 42, 8579.

76. Quinone Products from Bergman cycloaromatization – the role of molecular oxygen, Philip M. Warner and Graham B. Jones, Journal of Organic Chemistry,  2001, 66, 8859.

75. Butalene and Related Compounds- Aromatic or Antiaromatic?, Philip M. Warner and Graham B. Jones, Journal of the American Chemical Society, 2001, 123, 10322.

74. Bidendate Planar Chiral (6-Arene Tricarbonyl Chromium(0) Complexes: Ligands for Catalytic Asymmetric Alkene Hydrosilylation, Weber, I. ; Jones, G. B. Tetrahedron Lett. 2001, 42, 6983.

73. Shielding in Organic Synthesis, Graham B. Jones, Tetrahedron, 2001, 57, 7999.

72. Quinone Isomers of the WS-5995 Antibiotics: Synthetic Antitumor Agents that Inhibit Macromolecule Synthesis, Elisabeth M. Perchellet, Bonnie Sperfslage,  Ghassan Qabaja, Graham B. Jones, Jean-Pierre Perchellet,  Anti-Cancer Drugs, 2001, 12, 401.

71. Electronic Control of the Bergman Cyclization: The Remarkable Role of Vinyl Substitution, Graham B. Jones and Philip M. Warner, Journal of the American Chemical Society, 2001, 123, 2134.

70. Target Directed Enediynes: Designed Estramycins, Graham B. Jones, George Hynd, Justin M. Wright, Gary W. Plourde II, Robert S. Huber, Jude E. Mathews, Aiwen Li, Michael W. Kilgore, Molly Yancisin, and Myles Brown, Journal of Organic Chemistry2001, 66, 3688.

69. Enantioselective Catalysis using Planar Chiral h6 Arene Chromium Complexes: 1,2-Diols as Cycloaddition Catalysts, Graham B. Jones, Mustafa Guzel, and Steven B. Heaton, Tetrahedron: Asymmetry 2000, 11, 4303.

68. Annulation Strategies in Benzo[b]quinone Synthesis: Efficient Routes to Kinafluorenone and the WS-599A Antibiotics, Ghassan Qabaja, and Graham B. Jones, Journal of Organic Chemistry, 2000, 65, 7187.

67. Synthesis and Photochemical Activity of Designed Enediynes, Graham Jones, Justin Wright, Gary Plourde II, Ajay D. Purohit, Justin Wyatt, George Hynd, and Farid Fouad, Journal of the American Chemical Society, 2000, 122, 9872.

66. An Enzyme Activated Antiprostatic Prodrug, Graham B. Jones, Miguel O. Mitchell, James S. Weinberg, Anthony V. D’Amico, Glenn A. Bubley, Bioorganic and Medicinal Chemistry Letters, 2000, 10, 1987.

65. An Intramolecular Arylation Route to the Kinafluorenones, Ghassan Qabaja, Graham B. Jones, Tetrahedron Letters, 2000, 41, 5317.

64. Protein-Degrading Enediynes: Library Screening of Bergman Cycloaromatization Products, Graham B. Jones, Justin M. Wright, George Hynd, Justin K. Wyatt, Molly Yancisin, and Myles A. Brown Organic Letters, 2000, 2, 1863.

63. Electronic Control of the Bergman Cycloaromatization: Synthesis and Chemistry of Chloroenediynes, Jones, G. B. ; Plourde, G. W.  Organic Letters,  2000, 2, 1757.

62. Exploiting p Shielding Interactions in a h6 Arene Complexed Chiral Auxiliary, Graham B. Jones and Mustafa Guzel, Tetrahedron Letters, 2000, 41, 4695.

61. Catalytic Enantioselective Cycloadditions:  A Readily Available Diels-Alder Catalyst, Graham B. Jones and Mustafa Guzel, Tetrahedron: Asymmetry, 2000, 11, 1267.

60. Regioselective Lactonization of Naphthoquinones:  Synthesis and Antitumoral Activity of the WS 5995 Antibiotics, Ghassan Qabaja, Elisabeth M. Perchellet, Jean-Pierre Perchellet and Graham B. Jones, Tetrahedron Letters, 2000, 41, 3007.

59. Understanding Enediyne-Protein Interactions: Diyl Atom Transfer Results in Generation of Aminoacyl Radicals” Jones, G. B. ; Plourde, G. W. ; Wright, J. M. ; Organic Letters, 2000, 2, 811.

58. A Direct and Stereocontrolled Route to Conjugated Enediynes, Graham B. Jones, Justin M. Wright,Gary W. Plourde II, George Hynd, Robert S. Huber, and Jude E. Mathews, Journal of the American Chemical Society, 2000, 122, 1937.

57. Stereoselective Route to Mitosanes via Tricarbonyl h6 Arene Chromium Complexes, Graham Jones, Mustafa Guzel, and Jude E. Mathews, Tetrahedron Letters, 2000, 41, 1123.

56. On the Selective Deprotection of Trityl Ethers, Jones, G. B. ; Hynd, G. ; Wright, J. W. ; Sharma, A. , Journal of Organic Chemistry,  2000, 65, 263.

55. Synthesis and DNA Binding of Spirocyclic Model Compounds Related to the Neocarzinostatin Chromophore, Xi, Z.; Jones, G. B. ; Qabaja, G. ;  Wright, J. W. ;  Johnson, F. S. ;  Goldberg, I. H. ; Org. Lett. 1999, 1, 1375.

54. Stereoselective access to Substituted Enediyne Building Blocks, Hynd, G. ; Jones, G. B. ; Plourde, G. W. ; Wright, J. W. ; Tetrahedron Lett. 1999, 40, 4481.

53. Stereochemical control in the metallohalocarbenoid route to linear enediynes, Wright, J. W. ; Jones, G. B. ; Tetrahedron Lett. 1999, 40, 7605.

52. Tricarbonyl (h6 arene) Chromium (0) Complexes Derived from 8-Phenylmenthol Chiral Auxiliaries, William T. Pennington, Brant J. Chapman, and Graham B. Jones, J. Chem. Cryst. 1999, 5455.

51. Mixed Ligand Arene Chromium Carbonyl Complexes as Electronic Modulators, G. B. Jones, B. J. Chapman, and J. E. Mathews, J. Org. Chem.,  1998, 63, 2928.

50. Enediyne Hybrids in Chemotherapeutic and Chemopreventative Pathways, Intl. J. Modern Cancer Therapy., 1998, 1, 1.

49. Enantioselective Cycloadditions Catalyzed by Face Resolved Arene Chromium Carbonyl Complexes, Graham B. Jones and Mustafa Guzel, Tetrahedron: Asymmetry, 1998, 9, 2023.

48. Refined Enantioselective Methylation Catalysts: Improved Routes to Bifunctional C5 Synthons, Graham B. Jones, Mustafa Guzel and Brant J. Chapman, Tetrahedron: Asymmetry, 1998, 9, 901.

47. Cancer Chemotherapy: From Mustard Gas to Medicines, Chem. Heritage, 1998, 15(2), 8.

46. On the Origins of Enantioselectivity in Oxazaborolidine Mediated Carbonyl Reductions, Graham B. Jones, Steven B. Heaton, Mustafa Guzel, and Brant J. Chapman, Tetrahedron: Asymmetry, 1997, 8, 3625.

45. Facile Unmasking of Dicobalt Hexacarbonyl Complexes of 1-Cyclodecen-3,9-diynes [Enediynes], Graham B. Jones, Justin M. Wright, Teresa  M. Rush, Gary W. Plourde II, Thomas F. Kelton, Jude E. Mathews, Robert S. Huber and James P. Davidson J. Org. Chem.,  1997, 62, 9379.

44. Bifunctional Antitumor Agents.  Derivatives of Pyrrolo[9, 10-b]phenanthrene- an Intercalative Prodrug Delivery Template, G. B. Jones and J. E. Mathews, Tetrahedron, 1997, 53, 14599.

43. Catalytic Enantioselective Synthesis of Macrolides via Asymmetric Alkylation, G. B. Jones, R. S. Huber and B. J. Chapman, Tetrahedron: Asymmetry, 1997, 8, 1797.

42. Bifunctional Antitumor Agents: A DNA Interactive Enediyne from the Pyrrolophenanthrene Template, G. B. Jones and J. E. Mathews, Bioorg. Med. Chem. Lett., 1997, 7, 745.

41.  p Stacking Effects: Can They Be Modulated? Graham B. Jones and Brant J. Chapman, Synlett, 1997, 439.

40. Jones, G. B. ; Chapman, B. J. ; Phenylethynylcopper(I), in Encyclopedia of Reagents for Organic Synthesis: Paquette, L. A. , Ed; Wiley, New York, 1996.

39. Jones, G. B. ; Chapman, B. J. ; Phenylethynylcopper(I)-Tris(tributylphosphine), in Encyclopedia of Reagents for Organic Synthesis: Paquette, L. A. , Ed; Wiley, New York, 1996.

38. Jones, G. B. ; Chapman, B. J. ; (Trimethylsilyl)ethynylcopper(I), in Encyclopedia of Reagents for Organic Synthesis: Paquette, L. A. , Ed; Wiley, New York, 1996.

37. Jones, G. B. ; Chapman, B. J. ; Hexynylcopper, in Encyclopedia of Reagents for Organic Synthesis: Paquette, L. A. , Ed; Wiley, New York, 1996.

36. Jones, G. B. ; Chapman, B. J. ; Methoxy-3-methylbutynylcopper, in Encyclopedia of Reagents for Organic Synthesis: Paquette, L. A. , Ed; Wiley, New York, 1996.

35. Jones, G. B. ; Chapman, B. J. ; Pentynylcopper, in Encyclopedia of Reagents for Organic Synthesis: Paquette, L. A. , Ed; Wiley, New York, 1996.

34. Jones, G. B. ; Chapman, B. J. ; 1-Pentynylcopper(I)-Hexamethylphosphoric Triamide, in Encyclopedia of Reagents for Organic Synthesis: Paquette, L. A. , Ed; Wiley, New York, 1996.

33. Jones, G. B. ; Chapman, B. J. ; (Trimethylsilyl)propynylcopper(I), in Encyclopedia of Reagents for Organic Synthesis: Paquette, L. A. , Ed; Wiley, New York, 1996.

32. Jones, G. B. ; Chapman, B. J. ; Copper(I)isoprenylacetylide, in Encyclopedia of Reagents for Organic Synthesis: Paquette, L. A. , Ed; Wiley, New York, 1996.

31. Jones, G. B. ; Chapman, B. J. ; Chlorodiiodomethane, in Encyclopedia of Reagents for Organic Synthesis: Paquette, L. A. , Ed; Wiley, New York, 1996.

30. Jones, G. B. ; Huber, R. S. ; 1,1 Carbonyl bis(3-methylimidazolium)triflate, in Encyclopedia of Reagents for Organic Synthesis: Paquette, L. A. , Ed; Wiley, New York, 1996.

29. Jones, G. B. ; Chapman, B. J. ; Cyclopentadienone diethyl  acetal, in Encyclopedia of Reagents for Organic Synthesis: Paquette, L. A. , Ed; Wiley, New York, 1996.

28. Target Directed Enediyne Prodrugs: hER and AhR Degradation by a Synthetic Oxo-Enediyne, Graham B. Jones, Michael W. Kilgore, Richard S. Pollenz, Aiwen Li, Jude E. Mathews, Justin M. Wright, Robert S. Huber, Patricia L. Tate, Thomas L. Price, and Robert P. Sticca, Bioorg. Med. Chem. Lett., 1996, 6, 1971.

27. Jones, G. B. ; Chapman, B. J. ; Pyrroles and their Benzo Derivatives:Structure, in Comprehensive Heterocyclic Chemistry II; Pergamon, Oxford, 1996, pp. 1-38.

26. Target Directed Enediyne Prodrugs: Cytotoxic Estrogen Conjugates, Graham B. Jones, Robert S. Huber, Jude E. Mathews and Aiwen Li, Tetrahedron Lett., 1996, 37, 3643.

25. Jones, G. B. ; Mathews, J. E. ; Synthesis of Carbon Atoms Bearing Halogens and Heteroatoms, in Organic Functional Group Transformations; Katritzky, A. R. ; Rees, C. W. ; Meth-Cohn, O. ; Eds; Pergamon, Oxford, 1995, pp. 35-66.

24. Towards Enediyne Libraries: Cyclic Enediynes via an Intramolecular Carbenoid Coupling Protocol; Graham B. Jones, Robert S. Huber and Jude E. Mathews, J. Chem. Soc. Chem. Commun., 1995, 1791.

23. p Stacking Effects in Organic Synthesis; Graham B. Jones and Brant J. Chapman, Synthesis, 1995, 475.

22. Tricarbonyl h6 Arene Chromium (0) Based Antitumor Agents, Graham B. Jones and Jude E. Mathews , Bioorg. Med. Chem. Lett., 1995, 5, 93.

21. Catalytic Enantioselective Macrolide Synthesis II: Use of Differential Deprotection Protocols; Graham B. Jones, Brant J. Chapman, Robert S. Huber and Reeshemah Beaty; Tetrahedron: Asymmetry, 1994, 5, 1199.

20. Adenylated Dinucleotide Binding to the Adenosine 5′,5”’Tetraphosphate Mouse Heart Receptor; R. H. Hilderman, J. E. Lilien, J. K. Zimmerman, D. H. Tate, M. A. Dimmick and G. B. Jones;  Biochem. Biophys. Res. Commun., 1994, 200, 749.

19. A Mild and Efficient Route to the Pharmacophore of the Enediyne Antitumor Agents – (Z)-1,6-[Bis (trimethylsilyl)]-Hex-3-ene-1,5-diyne via a Novel Carbenoid Coupling Reaction; Graham B. Jones and Robert S. Huber, Tetrahedron Lett., 1994, 35, 2655.

18. Pyrrolo [9, 10] phenanthrenes: Versatile Intercalative Drug Delivery Vehicles, Graham B. Jones, Jude E. Mathews and W. Kenneth Banner, Heterocycles, 1994, 38, 1221.

17. Decarboxylation of Indole-2-Carboxylates: Improved Procedures; Graham B. Jones and Brant J. Chapman,  J. Org. Chem., 1993, 58, 5558.

16. The First Catalytic Enantioselective Synthesis of (R)-Lasiodiplodin; Graham B. Jones and Robert S. Huber, Synlett, 1993, 367.

15. Catalytic Asymmetric Induction II. Highly Selective 1,2 Alkyl Additions to Aldehydes using Chiral Arene Chromium Tricarbonyl Complexes as Enantioselective Catalysts; Steven B. Heaton and Graham B. Jones, Tetrahedron: Asymmetry, 1993, 4, 261.

14. Preparation of Tricarbonyl (h6 arene) Chromium (0) Complexes Derived from (S)-2-Indoline Carboxylic Acid; Steven B. Heaton, Graham B. Jones and William T. Pennington, Acta Crystallographica, 1993, C49, 1749.

13. The Claisen Rearrangement in Synthesis: Acceleration of the Johnson Orthoester Protocol en route to Bicyclic Lactones;  Graham B. Jones, Robert S. Huber and Sotheary Chau, Tetrahedron, 1993, 49, 369.

12. Acceleration of the Orthoester Claisen Rearrangement by Clay Catalyzed Microwave Thermolysis: Expeditious Route to Bicyclic Lactones; Robert S. Huber and Graham B. Jones,  J. Org. Chem., 1992, 57, 5778.

11. Chiral Arene Chromium Tricarbonyl Complexes as Enantioselective Catalysts: Highly Selective 1,2 Alkyl Additions to Aldehydes; Steven B. Heaton and Graham B. Jones, Tetrahedron Lett., 1992, 33, 1693.

10. Reductive Cleavage of tert-Butyldimethylsilyl Ethers by Diisobutylaluminum Hydride”; E. J. Corey and Graham B. Jones, J. Org. Chem., 1992, 57, 1028.

9. Enantioselective Route to a-Hydroxy Aldehyde and Acid Derivatives; E. J. Corey and Graham B. Jones, Tetrahedron Lett., 1991, 32, 5713.

8. Cyclopropamitosenes, Novel Bioreductive Anticancer Agents. Synthesis of 7-Methoxycyclopropamitosene and Related Indolequinones; Ann S. Cotterill, Paul Hartopp, Graham B. Jones, Christopher J. Moody, Claire L. Norton, Noleen O’Sullivan and Elizabeth Swann; Tetrahedron, 1994, 50, 7657.

7. Inter- and Intramolecular Reactions of 2-Indolyl Carbenes and Related Species. Preparation of 1,2- Aziridinopyrrolo[1,2-a]indoles; Graham B. Jones, Christopher J. Moody, Albert Padwa and Jamal M. Kassir, J.  Chem.  Soc.,  Perkin Trans. 1., 1991, 1721.

6. Structurally Modified Antitumour Agents part 2. Total Synthesis of a Cyclopropamitosene; Graham B. Jones and Christopher J. Moody, J.  Chem.  Soc.,  Perkin Trans. 1., 1989, 2455.

5. Structurally Modified Antitumour Agents part 1. Synthesis of Cyclopropapyrrolo[1,2a]indoles Related to Mitosenes by Intramolecular Cycloaddition; Graham B. Jones and Christopher J. Moody, J. Chem. Soc., Perkin Trans. 1., 1989, 2449.

4. Structurally Modified Antitumour Agents – Synthesis of a Cyclopropamitosene; Graham B. Jones and Christopher J. Moody, J.  Chem.  Soc., Chem.  Commun., 1989, 186.

3. Fused Aziridines via Intramolecular Cycloaddition;  Graham B. Jones and Christopher J. Moody, J.  Chem.  Soc., Chem.  Commun. , 1988, 1009.

2. Cyclopropapyrrolo[1,2-a]indoles, Graham B. Jones and Christopher J. Moody; J. Chem. Soc., Chem. Commun., 1988, 166.

1. F.V.P. of 1 -Allylbenzotriazoles and Dihydrobenzoxazines: Formation of Quinolines; S. J. Barker, G. B. Jones, K. R. Randles and R. C. Storr, Tetrahedron Lett., 1988, 29, 953.

 

Books Edited

Advances in DNA Sequence Specific Agents, Volume 4, Elsevier, Amsterdam, 2002

Advances in DNA Sequence Specific Agents, Volume 3, JAI, Greenwich, 1998